Drug class and membersAction on affected neurotransmitterNeuroreceptors
AnticholinergicsAcetylcholine antagonistsNicotinic and muscarinic
Asthmador
Benztropine (Cogentin)
Dimenhydrinate (Dramamine)
Diphenhydramine (Benadryl)
Hydroxyzine (Atarax)
Locoweed
DissociativesAffect actions of all neurotransmittersAll receptors
Ketamine (Ketalar)
Phencyclidine (PCP)
Phenylcyclohexylpyrolidine (PHP)
Opiatesβ-Endorphin agonists
Butorphanol (Stadol)κ
Pentazocine (Talwin)
Heroinμ
Hydromorphone (Dilaudid-Hp)
Mesipramine
Methadone
Morphine
PsychedelicsSerotonin agonists5-HT-2
Borneol
Lysergic acid diethylamide (LSD)
Mescaline
Methylenedioxymeth-amphetamine (MDA)
Psilocybin
Sufrole
Sedative-hypnoticsGABA agonistsGABA-A
Barbiturates
Ethchlorvinyl (Placidyl)
Glutethimide (Doriden)
Methaqualone
Zolpidem (Ambien)
BenzodiazepinesGABA-A-α
Ethyl alcoholGABA and opioid agonistGABA-A and μ
StimulantsDopamine, norepinephrine and serotonin agonistsDA-2, 5-HT-2, α and β
Amphetamine
Cocaine
Methamphetamine (Desoxyn)
Methylphenidate (Ritalin)